BX517(PDK1 inhibitor2)
BX517
CAS: 850717-64-5
Molecular Formula: C15H14N4O2
BX517(PDK1 inhibitor2) - Names and Identifiers
BX517(PDK1 inhibitor2) - Physico-chemical Properties
| Molecular Formula | C15H14N4O2 |
| Molar Mass | 282.3 |
| Solubility | DMSO: ≥ 27 mg/mL |
| Storage Condition | -20℃ |
| In vitro study | BX-517 blocks activation of Akt in tumor cells, is potent with IC 50 of 0.1-1.0 μM. BX-517 blocks AKT2 activation in cells with submicromolar potency. BX-517 is 100-fold selective or better against a panel of seven additional Ser/Thr and Tyr kinases. |
BX517(PDK1 inhibitor2) - Preparation solution concentration reference
| 1mg | 5mg | 10mg | |
|---|---|---|---|
| 1 mM | 3.542 ml | 17.712 ml | 35.424 ml |
| 5 mM | 0.708 ml | 3.542 ml | 7.085 ml |
| 10 mM | 0.354 ml | 1.771 ml | 3.542 ml |
| 5 mM | 0.071 ml | 0.354 ml | 0.708 ml |
Last Update：2024-01-02 23:10:35
BX517(PDK1 inhibitor2) - Reference Information
| biological activity | BX517 is a potent, selective PDK1 inhibitor with an IC50 value of 6 nM. |
| Target | IC50: 6 nM (PDK1) |
Last Update：2024-04-09 02:00:14
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Product Name: BX517 Visit Supplier Webpage Request for quotation
CAS: 850717-64-5
Tel: 18301782025
Email: 3008007409@qq.com
Mobile: 18021002903
QQ: 3008007409
Wechat: 18301782025
CAS: 850717-64-5
Tel: 18301782025
Email: 3008007409@qq.com
Mobile: 18021002903
QQ: 3008007409
Wechat: 18301782025
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